Published 06 Jan 2020
Beilstein Arch. 2020, 20203. doi:10.3762/bxiv.2020.3.v1
Published 05 Dec 2019
Beilstein Arch. 2019, 2019152. doi:10.3762/bxiv.2019.152.v1

Synthesis and herbicidal activity of aryloxyacetic acid derivatives as HPPD inhibitors

  • Man-Man Wang,
  • Hao Huang,
  • Lei Shu,
  • Jian-Min Liu,
  • Jian-Qiu Zhang,
  • Yi-Le Yan and
  • Da-Yong Zhang
Published 28 Nov 2019
Beilstein Arch. 2019, 2019150. doi:10.3762/bxiv.2019.150.v1

Syntheses of xanthone derivatives and their bioactivity investigation

  • Beidou Zhou,
  • Zhimin Weng,
  • Yugui Tong,
  • Zetong Ma,
  • Rongrong Wei,
  • Jiali Li and
  • Zihan Yu
Published 27 Nov 2019
Beilstein Arch. 2019, 2019148. doi:10.3762/bxiv.2019.148.v1
Published 19 Nov 2019
Beilstein Arch. 2019, 2019146. doi:10.3762/bxiv.2019.146.v1

NOVEL COMPOUNDS FROM CONDENSATION REACTION BETWEEN 2-ACETYLPYRIDINE AND 2-FORMYLPYRIDINE. SYNTHESIS, CRYSTAL STRUCTURE AND BIOLOGICAL EVALUATION

  • Roman Vasile Rusnac,
  • Maria Stefan Botnaru,
  • Nicanor Barba,
  • Peter Alexei Petrenko,
  • Yurii Chumakov and
  • Aurelian Petru Gulea
Published 18 Nov 2019
Beilstein Arch. 2019, 2019145. doi:10.3762/bxiv.2019.145.v1

Practical method to obtain α-acetoxyketones promoted by (diacetoxyiodo)benzene and acetic acid

  • Osvaldo J Quintana-Romero,
  • Jorge Camacho-Ruiz and
  • Armando Ariza-Castolo
Published 13 Nov 2019
Beilstein Arch. 2019, 2019144. doi:10.3762/bxiv.2019.144.v1

Synthesis and cytotoxicity of novel oxindoles dispiro derivatives with thiohydantoin and adamantane fragments

  • Maxim E. Kukushkin,
  • Dmitriy A. Skvortsov,
  • Marina A. Kalinina,
  • Viktor A. Tafeenko,
  • Vladimir V. Burmistrov,
  • Gennady M. Butov,
  • Nikolai V. Zyk,
  • Alexander G. Majouga and
  • Elena K. Beloglazkina
Published 11 Nov 2019
Beilstein Arch. 2019, 2019143. doi:10.3762/bxiv.2019.143.v1

Efficient Method for Propargylation of Aldehydes Promoted by Allenyl Boron Compounds under Microwave Irradiation

  • Jucleiton JR Freitas,
  • Queila PSB Freitas,
  • Silvia RCP Andrade,
  • Juliano CR Freitas,
  • Roberta A Oliveira and
  • Paulo H Menezes
Published 01 Nov 2019
Beilstein Arch. 2019, 2019138. doi:10.3762/bxiv.2019.138.v1

Microwave-assisted Synthesis of 2-Substituted 4,5,6,7-Tetrahydro-1,3-thiazepines from 4-Aminobutanol

  • María C. Mollo,
  • Natalia B. Kilimciler,
  • Juan A. Bisceglia and
  • Liliana R. Orelli
Published 28 Oct 2019
Beilstein Arch. 2019, 2019135. doi:10.3762/bxiv.2019.135.v1
Published 28 Oct 2019
Beilstein Arch. 2019, 2019134. doi:10.3762/bxiv.2019.134.v1
Published 25 Oct 2019
Beilstein Arch. 2019, 2019131. doi:10.3762/bxiv.2019.131.v1
Published 24 Oct 2019
Beilstein Arch. 2019, 2019129. doi:10.3762/bxiv.2019.129.v1

Total synthesis of 2'-O-methyl-β-L-arabinosyluridine and reassignment the nucleoside from Penicillium sp. as 2'-O-methyl-β-L-uridine

  • chunyang shen,
  • Haixin Ding,
  • Xueping Tao,
  • Ruchun Yang,
  • Jiang Bai,
  • Banpeng Cao,
  • Yiyuan Peng and
  • Qiang Xiao
Published 23 Oct 2019
Beilstein Arch. 2019, 2019128. doi:10.3762/bxiv.2019.128.v1
Published 15 Oct 2019
Beilstein Arch. 2019, 2019121. doi:10.3762/bxiv.2019.121.v1

Synthesis, structural characterization and biological activity of new pyrazolo[4,3-e][1,2,4]triazine acyclonucleosides

  • Mariusz Mojzych,
  • Zbigniew Karczmarzyk,
  • Joanna Matysiak and
  • Andrzej Fruziński
Published 09 Sep 2019
Beilstein Arch. 2019, 2019102. doi:10.3762/bxiv.2019.102.v1
Published 03 Sep 2019
Beilstein Arch. 2019, 201998. doi:10.3762/bxiv.2019.98.v1
Published 28 Aug 2019
Beilstein Arch. 2019, 201992. doi:10.3762/bxiv.2019.92.v1

Unexpected one-pot formation of 1H-6a,8a-epiminotricyclopenta[a,c,e][8]annulene system from cyclopentanone, ammonia and dimethyl fumarate. Synthesis of highly strained polycyclic nitroxide and  EPR study

  • Sergey Dobrynin,
  • Igor Kirilyuk,
  • Yuri Gatilov,
  • Andrey Kuzhelev,
  • Olesya Krumkacheva,
  • Matvey Fedin,
  • Michael Bowman and
  • Elena Bagryanskaya
Published 20 Aug 2019
Beilstein Arch. 2019, 201987. doi:10.3762/bxiv.2019.87.v1

An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agent

  • Nicky J Willis,
  • Elliott D Bayle,
  • George Papageorgiou,
  • David Steadman,
  • Benjamin N Aktinson,
  • William Mahy and
  • Paul V Fish
Published 16 Jul 2019
Beilstein Arch. 2019, 201970. doi:10.3762/bxiv.2019.70.v1

Palladium-catalyzed Conia-ene Reaction of 1-alkynylindolin-3-ones: a strategy for the construction of Pyrrolo[1,2-a]indoles

  • Yong-Qin Tang,
  • Xing-Hai Fei,
  • Jian-Xiong An,
  • Fen-Fen Yang,
  • Dong-Zhu Duan,
  • Zuo-Xian Cao,
  • Xiao-Zhong Fu,
  • Yuan-Yong Yang,
  • Bin He and
  • Yong-Long Zhao
Published 04 Jul 2019
Beilstein Arch. 2019, 201959. doi:10.3762/bxiv.2019.59.v1

Synthesis of multi-substituted indene derivatives from aryl, vinyl, and alkyl/aryl carbinols

  • Mithun Chakraborty,
  • Gaddam Mahesh,
  • Omkar R. Nakel,
  • Gautamee Chavda,
  • Susarla Anusha and
  • Gangarajula Sudhakar
Published 07 Jun 2019
Beilstein Arch. 2019, 201939. doi:10.3762/bxiv.2019.39.v1

Synthesis of 1-azaspiro[4.4]nonan-1-oxyls via Intramolecular 1,3-Dipolar Cycloaddition

  • Yulia V. Khoroshunova,
  • Denis A. Morozov,
  • Andrey I. Taratayko,
  • Polina D. Gladkikh,
  • Yuri I. Glazachev and
  • Igor A. Kirilyuk
Published 03 Jun 2019
Beilstein Arch. 2019, 201937. doi:10.3762/bxiv.2019.37.v1

Installation of sulfonyl fluorides onto primary amides

  • Jing Liu,
  • Shi-Meng Wang and
  • Hua-Li Qin
Published 29 May 2019
Beilstein Arch. 2019, 201933. doi:10.3762/bxiv.2019.33.v1

Characterization of two new degradation products of atorvastatin-calcium formed upon treatment with strong acids

  • Jürgen Krauß,
  • Monika Klimt,
  • Markus Luber,
  • Peter Mayer and
  • Franz Bracher
Published 28 May 2019
Beilstein Arch. 2019, 201931. doi:10.3762/bxiv.2019.31.v1
OTHER BEILSTEIN-INSTITUT OPEN SCIENCE ACTIVITIES