The asymmetric Henry reaction as synthetic tool for production of drugs Linezolid and Rivaroxaban

  • Martin Vrbický,
  • Karel Macek,
  • Jaroslav Pochobradský,
  • Jan Svoboda,
  • Miloš Sedlák and
  • Pavel Drabina
Published 17 Jan 2022
Beilstein Arch. 2022, 20224. doi:10.3762/bxiv.2022.4.v1
Published 30 Nov 2021
Beilstein Arch. 2021, 202183. doi:10.3762/bxiv.2021.83.v1
Published 16 Aug 2021
Beilstein Arch. 2021, 202158. doi:10.3762/bxiv.2021.58.v1
Published 28 Jul 2021
Beilstein Arch. 2021, 202153. doi:10.3762/bxiv.2021.53.v1

Enantioselective PCCP Brønsted Acid Catalyzed Aminalization of Aldehydes

  • Martin Kamlar,
  • Robert Reiberger,
  • Martin Nigríni,
  • Ivana Císařová and
  • Jan Veselý
Published 28 Jun 2021
Beilstein Arch. 2021, 202148. doi:10.3762/bxiv.2021.48.v1
Published 25 May 2021
Beilstein Arch. 2021, 202140. doi:10.3762/bxiv.2021.40.v1

Copper-Mediated Oxidative C−H/N−H Activations with Alkynes by Removable Hydrazides

  • Feng Xiong,
  • Bo Li,
  • Chenrui Yang,
  • Liang Zou,
  • Wenbo Ma,
  • Linghui Gu,
  • Ruhuai Mei and
  • Lutz Ackermann
Published 21 May 2021
Beilstein Arch. 2021, 202139. doi:10.3762/bxiv.2021.39.v1

Unexpected synthesis and structure of a cage-like aza[3,3,3]propllane carbene

  • Ziqi Su,
  • Qi Zhang,
  • Guangwei Zhou,
  • Qianzhu Chen,
  • Yahan Xue,
  • Lizhu Zhang,
  • Qunsheng Yan,
  • Juan Xu,
  • Quansong Li and
  • Jiarong Li
Published 05 May 2021
Beilstein Arch. 2021, 202136. doi:10.3762/bxiv.2021.36.v1

Highly selective difluoromethylations of β-keto amides with TMSCF2Br under mild conditions

  • Yakun Wang,
  • Shuaifei Wang,
  • Conghui Zhang,
  • Ting Zhao,
  • Yanqin Hu,
  • Mingwei Zhang,
  • Pengli Chen,
  • Yang Fu and
  • Jieli Lv
Published 20 Apr 2021
Beilstein Arch. 2021, 202135. doi:10.3762/bxiv.2021.35.v1
Published 23 Mar 2021
Beilstein Arch. 2021, 202128. doi:10.3762/bxiv.2021.28.v1

DBU-catalyzed Michael addition of bulky glycine imine to α,β-unsaturated isoxazoles and pyrazolamides

  • Yu-Jun Bai,
  • Mei-Ling Cheng,
  • Xiao-Mu Hu,
  • Ya-Jun Bai,
  • Xiao-Hui Zheng,
  • Sheng-Yong Zhang and
  • Ping-An Wang
Published 09 Mar 2021
Beilstein Arch. 2021, 202118. doi:10.3762/bxiv.2021.18.v1
Published 08 Mar 2021
Beilstein Arch. 2021, 202117. doi:10.3762/bxiv.2021.17.v1
Published 25 Feb 2021
Beilstein Arch. 2021, 202114. doi:10.3762/bxiv.2021.14.v1

Metal-free visible-light-enabled vicinal trifluoromethyl dithiolation of unactivated alkenes

  • Xiaojuan Li,
  • Qiang Zhang,
  • Weigang Zhang,
  • Jinzhu Ma,
  • Yi Wang and
  • Yi Pan
Published 13 Jan 2021
Beilstein Arch. 2021, 20211. doi:10.3762/bxiv.2021.1.v1
Published 12 Nov 2020
Beilstein Arch. 2020, 2020129. doi:10.3762/bxiv.2020.129.v1
Published 09 Nov 2020
Beilstein Arch. 2020, 2020128. doi:10.3762/bxiv.2020.128.v1

Au(III) Complexes with tetradentate cyclam based ligands

  • Ann C Reiersølmoen,
  • Thomas N Solvi and
  • Anne Fiksdahl
Published 02 Nov 2020
Beilstein Arch. 2020, 2020124. doi:10.3762/bxiv.2020.124.v1
Published 26 Aug 2020
Beilstein Arch. 2020, 202097. doi:10.3762/bxiv.2020.97.v1

Mechanism of Base-Catalyzed Halogen Dance Reactions and the Role of Bromo-Bridged Transition States

  • Nader Sakhaee,
  • Yousef Fazaeli,
  • Esmail Doustkhah,
  • Sahar Sakhaee,
  • Ahmad Takallou and
  • Akbar Mobaraki
Published 27 Jul 2020
Beilstein Arch. 2020, 202086. doi:10.3762/bxiv.2020.86.v1

Ring closing metathesis of prochiral oxaenediynes to racemic 4-alkenyl-2-alkynyl-3,6-dihydro-2H-pyrans

  • Viola Kolaříková,
  • Markéta Rybáčková,
  • Martin Svoboda and
  • Jaroslav Kvíčala
Published 24 Jul 2020
Beilstein Arch. 2020, 202084. doi:10.3762/bxiv.2020.84.v1

Hierarchically assembled helicates as reaction platform – From stoichiometric Diels-Alder reactions to enamine catalysis

  • David Van Craen,
  • Jenny Begall,
  • Johannes Grosskurth,
  • Leonard Himmel,
  • Oliver Linnenberg,
  • Elisabeth Isaak and
  • Markus Albrecht
Published 17 Jul 2020
Beilstein Arch. 2020, 202082. doi:10.3762/bxiv.2020.82.v1
Published 09 Jun 2020
Beilstein Arch. 2020, 202070. doi:10.3762/bxiv.2020.70.v1

A Novel Sustainable Method to Prepare Glutaric Acid from Glucose

  • Lei Hao,
  • Chao Jie Li,
  • Lian Bo Zhao,
  • Xi Xian Xie and
  • Kui Lu
Published 19 May 2020
Beilstein Arch. 2020, 202062. doi:10.3762/bxiv.2020.62.v1
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