Halogenations of 3-aryl-1H-pyrazol-5-amines

  • Jing He,
  • Yueting Wei,
  • Yijiao Feng,
  • Chuntian Li,
  • Bin Dai and
  • Ping Liu
Published 24 Sep 2021
Beilstein Arch. 2021, 202166. doi:10.3762/bxiv.2021.66.v1

First Total Synthesis of Hoshinoamides A  

  • Haipin Zhou,
  • Zihan Rui,
  • Yiming Yang,
  • Shengtao Xu,
  • Yutian Shao and
  • Long Liu
Published 15 Sep 2021
Beilstein Arch. 2021, 202164. doi:10.3762/bxiv.2021.64.v1

Host-guest interaction and properties of cucurbit[8]uril with chloramphenicol

  • Lin Zhang,
  • Jun Zheng,
  • Guangyan Luo,
  • Xiaoyue Li,
  • Yunqian Zhang,
  • Zhu Tao and
  • Qianjun Zhang
Published 30 Aug 2021
Beilstein Arch. 2021, 202162. doi:10.3762/bxiv.2021.62.v1

Photophysical, photostability, and ROS generation properties of new trifluoromethylated quinoline-phenol Schiff bases

  • Inaiá O. Rocha,
  • Yuri G. Kappenberg,
  • Wilian C. Rosa,
  • Clarissa P. Frizzo,
  • Nilo Zanatta,
  • Marcos A. P. Martins,
  • Isadora Tisoco,
  • Bernardo A. Iglesias and
  • Helio G. Bonacorso
Published 23 Aug 2021
Beilstein Arch. 2021, 202160. doi:10.3762/bxiv.2021.60.v1

Reactivity of tetrazolo[1,5-a]pyrimidines in click chemistry and hydrogenation

  • Elisandra Scapin,
  • Geórgia C. Zimmer,
  • Jean C. B. Vieira,
  • Catarina A. B. Rodrigues,
  • Carlos A. M. Afonso,
  • Nilo Zanatta,
  • Helio G. Bonacorso,
  • Clarissa P. Frizzo and
  • Marcos A.P. Martins
Published 16 Aug 2021
Beilstein Arch. 2021, 202159. doi:10.3762/bxiv.2021.59.v1
Published 16 Aug 2021
Beilstein Arch. 2021, 202158. doi:10.3762/bxiv.2021.58.v1

Molecular rearrangement of pyrazino[2,3-c]quinolin-5(6H)-ones during their reaction with isocyanic acid

  • Antonín Klásek,
  • Antonín Lyčka,
  • Filip Křemen,
  • Aleš Růžička and
  • Michal Rouchal
Published 29 Jul 2021
Beilstein Arch. 2021, 202154. doi:10.3762/bxiv.2021.54.v1
Published 28 Jul 2021
Beilstein Arch. 2021, 202153. doi:10.3762/bxiv.2021.53.v1
Published 21 Jul 2021
Beilstein Arch. 2021, 202152. doi:10.3762/bxiv.2021.52.v1

Synthesis of new pyrazolo[1,2,3]triazines by cyclative cleavage of pyrazolyltriazenes

  • Nicolai Wippert,
  • Martin Nieger,
  • Claudine Herlan,
  • Nicole Jung and
  • Stefan Bräse
Published 13 Jul 2021
Beilstein Arch. 2021, 202151. doi:10.3762/bxiv.2021.51.v1

Ensemble-based virtual screening of Mycobacterium tuberculosis ClpC1 inhibitors

  • Hafsa Tayyab,
  • Nor F. W. Ridzwan and
  • Saharuddin B. Mohamad
Published 06 Jul 2021
Beilstein Arch. 2021, 202150. doi:10.3762/bxiv.2021.50.v1

Synthesis of 5-arylacetylene 1,2,4-oxadiazoles and their transformations under superelectrophilic activation conditions

  • Andrey I. Puzanov,
  • Dmitry S. Ryabukhin,
  • Anna S. Zalivatskaya,
  • Dmitriy N. Zakusilo,
  • Darya S. Mikson,
  • Irina A. Boyarskaya and
  • Aleksander Vasilyev
Published 30 Jun 2021
Beilstein Arch. 2021, 202149. doi:10.3762/bxiv.2021.49.v1

Enantioselective PCCP Brønsted Acid Catalyzed Aminalization of Aldehydes

  • Martin Kamlar,
  • Robert Reiberger,
  • Martin Nigríni,
  • Ivana Císařová and
  • Jan Veselý
Published 28 Jun 2021
Beilstein Arch. 2021, 202148. doi:10.3762/bxiv.2021.48.v1

Phenylamino pyrimidine-1,2,3-triazole derivatives as analogs of imatinib: searching for novel compounds against chronic myeloid leukemia

  • Luiz Claudio Ferreira Pimentel,
  • Lucas Villas Boas Hoelz,
  • Henayle Fernandes Canzian,
  • Frederico Silva Castelo Branco,
  • Andressa Paula de Oliveira,
  • Vinicius Rangel Campos,
  • Floriano Paes Silva Júnior,
  • Rafael Ferreira Dantas,
  • Jackson Antônio Lamounier Camargos Resende,
  • Anna Claudia Cunha,
  • Nubia Boechat and
  • Mônica Macedo Bastos
Published 09 Jun 2021
Beilstein Arch. 2021, 202144. doi:10.3762/bxiv.2021.44.v1

Synthesis and synthetic applications of (4-hydroxyphenyl)perfluoroalkylmethanols

  • Kyu Terashima,
  • Tomoko Kawasaki-Takasuka,
  • Ichiro Minami and
  • Takashi Yamazaki
Published 01 Jun 2021
Beilstein Arch. 2021, 202141. doi:10.3762/bxiv.2021.41.v1
Published 25 May 2021
Beilstein Arch. 2021, 202140. doi:10.3762/bxiv.2021.40.v1

Copper-Mediated Oxidative C−H/N−H Activations with Alkynes by Removable Hydrazides

  • Feng Xiong,
  • Bo Li,
  • Chenrui Yang,
  • Liang Zou,
  • Wenbo Ma,
  • Linghui Gu,
  • Ruhuai Mei and
  • Lutz Ackermann
Published 21 May 2021
Beilstein Arch. 2021, 202139. doi:10.3762/bxiv.2021.39.v1

Synthesis of halogenated bicyclic molecules involving Prins cyclization from aldehydes and non-conjugated diene alcohol

  • Kouichi Matsumoto,
  • Keisuke Ohtsuka,
  • Naruto Hasebe,
  • Kota Terada,
  • Masahiko Maekawa,
  • Yoshihide Nakao,
  • Keiji Nishiwaki and
  • Hideo Ando
Published 21 May 2021
Beilstein Arch. 2021, 202138. doi:10.3762/bxiv.2021.38.v1

Design and synthesis of highly oxygenated furo[3,2-c]pyran-4-ones and furo[3,2-c]chromen-4-ones scaffold as potential anticancer and antimicrobial agent

  • Suman Rani,
  • Nisha Kamra,
  • Sumit Thakral,
  • Devinder Kumar,
  • Ajeet Singh,
  • Payare L Sangwan and
  • Shashank K Singh
Published 17 May 2021
Beilstein Arch. 2021, 202137. doi:10.3762/bxiv.2021.37.v1

Unexpected synthesis and structure of a cage-like aza[3,3,3]propllane carbene

  • Ziqi Su,
  • Qi Zhang,
  • Guangwei Zhou,
  • Qianzhu Chen,
  • Yahan Xue,
  • Lizhu Zhang,
  • Qunsheng Yan,
  • Juan Xu,
  • Quansong Li and
  • Jiarong Li
Published 05 May 2021
Beilstein Arch. 2021, 202136. doi:10.3762/bxiv.2021.36.v1

Highly selective difluoromethylations of β-keto amides with TMSCF2Br under mild conditions

  • Yakun Wang,
  • Shuaifei Wang,
  • Conghui Zhang,
  • Ting Zhao,
  • Yanqin Hu,
  • Mingwei Zhang,
  • Pengli Chen,
  • Yang Fu and
  • Jieli Lv
Published 20 Apr 2021
Beilstein Arch. 2021, 202135. doi:10.3762/bxiv.2021.35.v1
Published 14 Apr 2021
Beilstein Arch. 2021, 202133. doi:10.3762/bxiv.2021.33.v1
Published 06 Apr 2021
Beilstein Arch. 2021, 202131. doi:10.3762/bxiv.2021.31.v1
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