Published 25 Feb 2021
Beilstein Arch. 2021, 202114. doi:10.3762/bxiv.2021.14.v1

Total Synthesis of Pyrrolo[2,3-c]quinoline Alkaloid: Trigonoine B

  • Takashi Nishiyama,
  • Erina Hamada,
  • Daishi Ishii,
  • Yuuto Kihara,
  • Nanase Choshi,
  • Natsumi Nakanishi,
  • Mari Murakami,
  • Kimiko Taninaka,
  • Noriyuki Hatae and
  • Tominari Choshi
Published 26 Jan 2021
Beilstein Arch. 2021, 20216. doi:10.3762/bxiv.2021.6.v1

Metal-free visible-light-enabled vicinal trifluoromethyl dithiolation of unactivated alkenes

  • Xiaojuan Li,
  • Qiang Zhang,
  • Weigang Zhang,
  • Jinzhu Ma,
  • Yi Wang and
  • Yi Pan
Published 13 Jan 2021
Beilstein Arch. 2021, 20211. doi:10.3762/bxiv.2021.1.v1

β-Lactamase inhibition profile of new amidine substituted diazabicyclooctanes

  • zafar iqbal,
  • Yuanyu Gao,
  • Dong Tang,
  • Xueqin Ma,
  • Jinbo Ji,
  • Jian Sun,
  • Jingwen Ji,
  • Yuanbai Liu,
  • Lijuan Zhai,
  • Rui Jiang,
  • Yangxiu Mu,
  • Lili He,
  • Haikang Yang and
  • Zhixiang Yang
Published 21 Dec 2020
Beilstein Arch. 2020, 2020143. doi:10.3762/bxiv.2020.143.v1

Synthesis of β-triazolylenones via metal-free desulfonylative alkylation of N-tosyl-1,2,3-triazoles

  • Soumyaranjan Pati,
  • Renata G. Almeida,
  • Eufrânio N. da Silva Júnior and
  • Irishi N. N. Namboothiri
Published 27 Nov 2020
Beilstein Arch. 2020, 2020134. doi:10.3762/bxiv.2020.134.v1

Synthesis of 1-Indolyl-3,5,8-Substituted γ-Carbolines: One Pot Metal-Solvent Free Protocol and Biological Evaluation

  • Premansh Dudhe,
  • Mena Asha Krishnan,
  • Kratika Yadav,
  • Diptendu Roy,
  • Krishnan Venkatasubbaiah,
  • Biswarup Pathak and
  • Venkatesh Chelvam
Published 19 Nov 2020
Beilstein Arch. 2020, 2020131. doi:10.3762/bxiv.2020.131.v1
Published 12 Nov 2020
Beilstein Arch. 2020, 2020129. doi:10.3762/bxiv.2020.129.v1
Published 09 Nov 2020
Beilstein Arch. 2020, 2020128. doi:10.3762/bxiv.2020.128.v1

A Column-Free and Aqueous Waste-Free Process for Thioamide Preparation with Lawesson’s reagent

  • Ke Wu,
  • Yichen Ling,
  • An Ding,
  • Liqun Jin,
  • Nan Sun,
  • Baoxiang Hu,
  • Zhenlu Shen and
  • Xinquan Hu
Published 05 Nov 2020
Beilstein Arch. 2020, 2020126. doi:10.3762/bxiv.2020.126.v1

Au(III) Complexes with tetradentate cyclam based ligands

  • Ann C Reiersølmoen,
  • Thomas N Solvi and
  • Anne Fiksdahl
Published 02 Nov 2020
Beilstein Arch. 2020, 2020124. doi:10.3762/bxiv.2020.124.v1
Published 28 Oct 2020
Beilstein Arch. 2020, 2020123. doi:10.3762/bxiv.2020.123.v1

Mesoionic tetrazolium-5-aminides: Synthesis, Molecular and Crystal Structures, UV-Vis Spectra, and DFT Calculations

  • Vladislav A. Budevich,
  • Sergei V. Voitekhovich,
  • Alexander V. Zuraev,
  • Vadim E. Matulis,
  • Vitaly E. Matulis,
  • Alexander S. Lyakhov,
  • Ludmila S. Ivashkevich and
  • Oleg A. Ivashkevich
Published 22 Oct 2020
Beilstein Arch. 2020, 2020122. doi:10.3762/bxiv.2020.122.v1
Published 12 Oct 2020
Beilstein Arch. 2020, 2020118. doi:10.3762/bxiv.2020.118.v1

Metal-free synthesis of biarenes via photoextrusion in di(tri)arylphosphates

  • Hisham Qrareya,
  • Lorenzo Meazza,
  • Stefano Protti and
  • Maurizio Fagnoni
Published 28 Sep 2020
Beilstein Arch. 2020, 2020110. doi:10.3762/bxiv.2020.110.v1
Published 25 Aug 2020
Beilstein Arch. 2020, 202096. doi:10.3762/bxiv.2020.96.v1
Published 25 Aug 2020
Beilstein Arch. 2020, 202094. doi:10.3762/bxiv.2020.94.v1
Published 27 Jul 2020
Beilstein Arch. 2020, 202085. doi:10.3762/bxiv.2020.85.v1

Models of Necessity

  • Timothy Clark and
  • Martin G Hicks
Published 19 Jun 2020
Beilstein Arch. 2020, 202077. doi:10.3762/bxiv.2020.77.v1

Transformation of 2H-1,2,3-benzothiadiazine 1,1-dioxides variously substituted at the aromatic ring, via nucleophilic substitution and demethylation reactions

  • Imre Gyűjtő,
  • Márta Porcs-Makkay,
  • Ernák Ferenc Várda,
  • Gyöngyvér Pusztai,
  • Gábor Tóth,
  • Gyula Simig and
  • Balázs Volk
Published 16 Jun 2020
Beilstein Arch. 2020, 202073. doi:10.3762/bxiv.2020.73.v1
Published 10 Jun 2020
Beilstein Arch. 2020, 202071. doi:10.3762/bxiv.2020.71.v1
Published 22 May 2020
Beilstein Arch. 2020, 202063. doi:10.3762/bxiv.2020.63.v1

A Novel Sustainable Method to Prepare Glutaric Acid from Glucose

  • Lei Hao,
  • Chao Jie Li,
  • Lian Bo Zhao,
  • Xi Xian Xie and
  • Kui Lu
Published 19 May 2020
Beilstein Arch. 2020, 202062. doi:10.3762/bxiv.2020.62.v1
Published 08 May 2020
Beilstein Arch. 2020, 202060. doi:10.3762/bxiv.2020.60.v1
Published 05 May 2020
Beilstein Arch. 2020, 202057. doi:10.3762/bxiv.2020.57.v1

Tuneable access to indole, indolone and cinnoline derivatives from a common 1,4-diketone Michael acceptor

  • Dalel El-Marrouki,
  • Sabrina Touchet,
  • Abderrahmen Abdelli,
  • Hédi M'Rabet,
  • Mohamed Lotfi Efrit and
  • Philippe C. Gros
Published 27 Apr 2020
Beilstein Arch. 2020, 202056. doi:10.3762/bxiv.2020.56.v1
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