Indium-mediated Domino Lactonisation Approach towards Diastereoselective Synthesis of Pyrazole C-3 Linked Butyrolactones

  • Dr Shubham Sharma,
  • Dr Virender Singh,
  • Dr Manpreet Singh and
  • Dr Ashutosh Sharma
Published 19 Apr 2023
Beilstein Arch. 2023, 202315. doi:10.3762/bxiv.2023.15.v1
Published 04 Apr 2023
Beilstein Arch. 2023, 202310. doi:10.3762/bxiv.2023.10.v1
Published 03 Apr 2023
Beilstein Arch. 2023, 20239. doi:10.3762/bxiv.2023.9.v1
Published 31 Jan 2023
Beilstein Arch. 2023, 20236. doi:10.3762/bxiv.2023.6.v1

An Efficient Metal-free and Catalyst-free C-S/C-O Bond Formation Strategy: Synthesis of Pyrazole Conjugated Thioamides and Amides

  • Shubham Sharma,
  • Dharmender Singh,
  • Sunit Kumar,
  • Vaishali  ,
  • Rahul Jamra,
  • Naveen Banyal,
  • Deepika  ,
  • Chandi C Malakar and
  • Virender Singh
Published 28 Dec 2022
Beilstein Arch. 2022, 202292. doi:10.3762/bxiv.2022.92.v1
Published 23 Nov 2022
Beilstein Arch. 2022, 202288. doi:10.3762/bxiv.2022.88.v1

Novel spirocyclic scaffold accessed via tandem Claisen rearrangement – intramolecular Michael addition

  • Anastasia Vepreva,
  • Alexander Yanovich,
  • Dmitry Dar'in,
  • Grigory Kantin,
  • Alexander Bunev and
  • Mikhail Krasavin
Published 11 Oct 2022
Beilstein Arch. 2022, 202283. doi:10.3762/bxiv.2022.83.v1

Polycyclic High Density Cage Compounds via Cross Metathesis

  • Sambasivarao Kotha and
  • Usha Nandan Chaurasia
Published 07 Oct 2022
Beilstein Arch. 2022, 202282. doi:10.3762/bxiv.2022.82.v1

Design and Synthesis of Pyrene Containing Unusual α-Amino Acid Derivatives

  • Sambasivarao Kotha,
  • Vidyasagar Gaikwad and
  • Saima Ansari
Published 06 Oct 2022
Beilstein Arch. 2022, 202281. doi:10.3762/bxiv.2022.81.v1

Novel Bis-Triazole Scaffold Accessed via Two Tandem [3+2] Cycloaddition Events Including an Uncatalyzed, Room-Temperature Azide-Alkyne Click Reaction

  • Ksenia Malkova,
  • Andrey Bubyrev,
  • Vasilisa Krivovicheva,
  • Dmitry Dar'in,
  • Alexander Bunev and
  • Mikhail Krasavin
Published 30 Sep 2022
Beilstein Arch. 2022, 202280. doi:10.3762/bxiv.2022.80.v1
Published 22 Sep 2022
Beilstein Arch. 2022, 202275. doi:10.3762/bxiv.2022.75.v1

Rhodium-catalyzed intramolecular reductive aldol-type cyclization: Application for the synthesis of a chiral necic acid lactone

  • Motoyuki Isoda,
  • Kazuyuki Sato,
  • Kenta Kameda,
  • Kana Wakabayashi,
  • Ryota Sato,
  • Hideki Minami,
  • Yukiko Karuo,
  • Atsushi Tarui,
  • Kentaro Kawai and
  • Masaaki Omote
Published 16 Sep 2022
Beilstein Arch. 2022, 202272. doi:10.3762/bxiv.2022.72.v1

One-pot Double Annulations to Confer Diastereoselective Spirooxindole-pyrrolothiazoles

  • Juan Lu,
  • Bin Yao,
  • Desheng Zhan,
  • Zhuo Sun,
  • Yun Ji and
  • Xiaofeng Zhang
Published 14 Sep 2022
Beilstein Arch. 2022, 202271. doi:10.3762/bxiv.2022.71.v1

ULTRASOUND-ASSISTED GREEN SYNTHESES OF NOVEL PYRIMIDINE DERIVATIVES AND THEIR COMPARISON WITH CONVENTIONAL METHODS

  • Vergush A. Pivazyan,
  • Emma A. Ghazaryan,
  • Armen V. Karapetyan,
  • Roza S. Shainova,
  • Siranush V. Harutyunyan,
  • Asya S. Vorskanyan,
  • Aleksandr P. Yengoyan and
  • Tiruhi A. Gomktsyan
Published 16 Aug 2022
Beilstein Arch. 2022, 202267. doi:10.3762/bxiv.2022.67.v1
Published 05 Jul 2022
Beilstein Arch. 2022, 202259. doi:10.3762/bxiv.2022.59.v1

Synthesis of Protected Precursors of Chitin Oligosaccharides by Electrochemical Polyglycosylation of Thioglycosides

  • Md Azadur Rahman,
  • Kana Kuroda,
  • Hirofumi Endo,
  • Norihiko Sasaki,
  • Tomoaki Hamada,
  • Hiraku Sakai and
  • Toshiki Nokami
Published 04 Jul 2022
Beilstein Arch. 2022, 202258. doi:10.3762/bxiv.2022.58.v1

Facile and Diastereoselective Arylation of the Privileged 1,4-Dihydroisoquinolin-3(2H)-one Scaffold

  • Dmitry Dar'in,
  • Grigory Kantin,
  • Alexander Bunev and
  • Mikhail Krasavin
Published 20 Jun 2022
Beilstein Arch. 2022, 202250. doi:10.3762/bxiv.2022.50.v1
Published 13 Jun 2022
Beilstein Arch. 2022, 202249. doi:10.3762/bxiv.2022.49.v1
Published 07 Jun 2022
Beilstein Arch. 2022, 202244. doi:10.3762/bxiv.2022.44.v1
Published 31 May 2022
Beilstein Arch. 2022, 202240. doi:10.3762/bxiv.2022.40.v1
Published 30 May 2022
Beilstein Arch. 2022, 202239. doi:10.3762/bxiv.2022.39.v1
Published 27 May 2022
Beilstein Arch. 2022, 202238. doi:10.3762/bxiv.2022.38.v1

Novel one-pot synthesis of 2-thio-substituted-3-H-phenothiazin-3-ones driven by oxidation with sodium periodate

  • Herman H. Odens Jr.,
  • Jae Y. You,
  • Alexandria D. Gallimore,
  • Preston H. Palm,
  • Cameron W. Davis,
  • Josue M. Bahena,
  • Jeffrey S. Moser,
  • Mackenzie E. Smith and
  • Herman H. Odens
Published 13 May 2022
Beilstein Arch. 2022, 202236. doi:10.3762/bxiv.2022.36.v1
Published 12 May 2022
Beilstein Arch. 2022, 202235. doi:10.3762/bxiv.2022.35.v1
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